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1,3-Diazepine Derivatives: Strategies for Synthesis
Yohan Malki,
Dr. Ludovic T. Maillard,
Prof. Nicolas Masurier,
Yohan Malki
IBMM, Université de Montpellier, CNRS, ENSCM, Montpellier, France
Search for more papers by this authorDr. Ludovic T. Maillard
IBMM, Université de Montpellier, CNRS, ENSCM, Montpellier, France
Search for more papers by this authorCorresponding Author
Prof. Nicolas Masurier
IBMM, Université de Montpellier, CNRS, ENSCM, Montpellier, France
Search for more papers by this authorYohan Malki,
Dr. Ludovic T. Maillard,
Prof. Nicolas Masurier,
Yohan Malki
IBMM, Université de Montpellier, CNRS, ENSCM, Montpellier, France
Search for more papers by this authorDr. Ludovic T. Maillard
IBMM, Université de Montpellier, CNRS, ENSCM, Montpellier, France
Search for more papers by this authorCorresponding Author
Prof. Nicolas Masurier
IBMM, Université de Montpellier, CNRS, ENSCM, Montpellier, France
Search for more papers by this authorGraphical Abstract
The present review describes the methodologies reported for the synthesis of 1,3-diazepine derivatives. This heterocyclic moiety forms the core structure of many compounds with potent biological activities. Synthetic strategies by ring closure or ring transformation are discussed.
Abstract
The present review describes the methodologies reported for the synthesis of 1,3-diazepine derivatives. This heterocyclic moiety forms the core structure of many compounds with potent biological activities. Synthetic strategies by ring closure or ring transformation are discussed.
Conflict of interest
The authors declare no conflict of interest.
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